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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T17877 | VH032-cyclopropane-F | VHL ligand 3,E3 ligase Ligand 19,Phenolic VH101 | Others , Ligand for E3 Ligase |
VH032-cyclopropane-F (Phenolic VH101) is a VH032-based VHL ligand. VH032-cyclopropane-F can be connected to the ligand for protein by a linker to form PROTACs. PROTAC 1 is a partial degrader of SMARCA2 and SMARCA4. | |||
T7759 | Thalidomide-O-amido-C4-NH2 TFA | E3 ligase Ligand-Linker Conjugates 19 TFA,Cereblon Ligand-Linker Conjugates 6 TFA | E3 Ligase Ligand-Linker Conjugate |
Thalidomide-O-amido-C4-NH2 TFA (E3 ligase Ligand-Linker Conjugates 19 TFA) is a synthesized E3 ligase ligand-linker conjugate. | |||
T17928 | Lenalidomide-C5-NH2 | E3 ligase Ligand-Linker Conjugates 31,Cereblon Ligand-Linker Conjugates 19 | Others |
Lenalidomide-C5-NH2 is the Lenalidomide-based Cereblon ligand used in the recruitment of CRBN protein. Lenalidomide-C5-NH2 can be connected to the ligand for protein by a linker to form PROTACs[1]. | |||
T17818 | Thalidomide-O-amido-C4-NH2 | E3 Ligase Ligand-Linker Conjugates 19,Cereblon Ligand-Linker Conjugates 6 | Others |
Thalidomide-O-amido-C4-NH2 (Cereblon Ligand-Linker Conjugates 6) is a synthesized ligand-linker conjugate that combines a Thalidomide-based cereblon ligand with a linker. It functions as an E3 ligase ligand-linker conjug... |